Visible light-mediated photocatalytic bromination of 2-arylimidazo[1,2-a]pyridines using CBr4 as bromine source

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초록

The photocatalytic bromination of 2-arylimidazo[1,2-a]pyridines is described in this paper. This reaction uses the readily accessible and shelf-stable CBr4 as a bromine source. This photocatalytic system is shown to serve as a convenient and practical synthetic protocol for the preparation of 2-aryl-3-bromoimidazo[1,2-a]pyridines.

키워드

Brominationphotoredox reaction2-arylimidazo[12-a]pyridines3-bromoimidazo[12-a]pyridinesASYMMETRIC-SYNTHESISPHOTOREDOX CATALYSISANTIVIRAL ACTIVITYCOUPLING REACTIONIMIDAZOHETEROCYCLESIMIDAZOPYRIDINESTETRAHYDROQUINOLINESHALOGENATIONACTIVATIONINHIBITORS
제목
Visible light-mediated photocatalytic bromination of 2-arylimidazo[1,2-a]pyridines using CBr4 as bromine source
저자
Lee, Ju HuiJung, Hye ImKim, Dae Young
DOI
10.1080/00397911.2019.1691738
발행일
2020-01-17
유형
Article
저널명
Synthetic Communications
50
2
페이지
197 ~ 206